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大环内酯类化合物雷帕霉素(Rapamycin,Rap)为哺乳动物雷帕霉素靶蛋白(Mammalian Target ofRapamycin,mTOR)特异性阻断剂,通过抑制mTOR活性,导致其下游底物真核细胞翻译启始因子4E结合蛋白1(elF4E-binding protein 1,4E-BP1)和核糖
The macrolide compound Rapamycin (Rap) is a specific blocker of Mammalian Target of Rapamycin (mTOR), which inhibits mTOR activity and leads to its downstream substrate eukaryotic cells Translation initiation factor 4E binding protein 1 (elF4E-binding protein 1,4E-BP1) and ribose